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197

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
TP1809 TAT

HIV Protease Microbiology/Virology; Proteases/Proteasome
TAT 源自人免疫缺陷病毒的转录反式激活因子,是一种细胞穿透肽。它可以增加异源蛋白质的产量和溶解度。
T38514 PMEDAP

Others; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
PMEDAP 是有效的人类免疫缺陷病毒 (HIV) 复制抑制剂。它具有抗小鼠巨细胞病毒活性。它有效抑制莫罗尼鼠肉瘤病毒诱导的肿瘤形成和相关死亡率。
T12953 Sodium copper chlorophyllin B

Influenza Virus; HIV Protease Microbiology/Virology; Proteases/Proteasome
Sodium copper chlorophyllin B 对流感病毒和HIV 有抗病毒活性,IC50s 值都是 50 到 100 μM。
T16764 RN-18

HIV Protease Microbiology/Virology; Proteases/Proteasome
RN-18是 HIV-1 病毒感染因子的一种拮抗剂。
T15436 GSK2838232

HIV Protease Microbiology/Virology; Proteases/Proteasome
GSK2838232 是一种新型人类免疫病毒成熟抑制剂,抑制 HIV 逆转录酶活性。
T10111 3-Deazaadenosine hydrochloride

Others; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
3-Deazaadenosine hydrochloride 是 S-腺苷高半胱氨酸水解酶的抑制剂,Ki 值为 3.9 µM。 它具有抗炎、抗增殖和抗 HIV 活性。
T12715 Reverse transcriptase-IN-1

HIV Protease Microbiology/Virology; Proteases/Proteasome
Reverse transcriptase-IN-1 是一种二芳基苯并嘧啶类似物,是一种有效的 HIV-1 非核苷类逆转录酶抑制剂,IC50 为 13.7 nM。
T9063 Clathrin-IN-1

HIV Protease Microbiology/Virology; Proteases/Proteasome
Clathrin-IN-1 是一种网格蛋白抑制剂,可通过与网格蛋白的末端域相关联来抑制网格蛋白介导的内吞作用,有潜力用于抗癌的研究。
T6256 YYA-021

YYA 021

gp120/CD4; HIV Protease Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
YYA-021具有高抗HIV 活性和低细胞毒性,是一种抑制HIV 进入的小分子CD4模拟物,。
T16276 NBD-556

HIV Protease Microbiology/Virology; Proteases/Proteasome
NBD-556是一种 CD4 模拟物,识别 HIV-1 包膜蛋白 gp120 并诱导 gp120 重组,类似于 CD4 结合,可阻断 gp120-CD4 的相互作用。
T4665 Temsavir

BMS626529

HIV Protease Microbiology/Virology; Proteases/Proteasome
Temsavir (BMS626529) 是一种新型附着抑制剂,靶向 HIV-1 gp120 并阻止其与 CD4+ T 细胞结合。
T15210 Elsulfavirine

Elpida,VM-1500

HIV Protease Microbiology/Virology; Proteases/Proteasome
Elsulfavirine (VM-1500) 是一种 HIV-1 感染的逆转录酶抑制剂,也是抗 HIV 的新药。
T0836 Sulfadoxine

周效磺胺,磺胺多辛,Sulphadoxine

DHFR; HIV Protease; Antibiotic; Parasite; Autophagy Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology; Proteases/Proteasome
Sulfadoxine (Sulphadoxine) 是磺胺类化合物,常与pyrimethamine 结合起到抗疟疾作用。它抑制HIV 在外周血单核细胞中的复制。
T0457 Probenecid

Benemid,丙磺舒

HIV Protease; Antibacterial; TRP/TRPV Channel Membrane transporter/Ion channel; Microbiology/Virology; Proteases/Proteasome
Probenecid (Benemid) 是一种苯甲酸衍生物,具有抗高尿酸特性。它也是一种选择性瞬时受体电位香草酸受体通道 2 激动剂,还可抑制pannexin 1通道。
T8311 Obefazimod

ABX-464,ABX464

HIV Protease Microbiology/Virology; Proteases/Proteasome
Obefazimod (ABX-464) 是一种抗HIV 剂。它抑制受刺激的外周血单核细胞中的 HIV-1 复制,IC50值为 0.1 μM 至 0.5 μM。
T4493 Bictegravir

GS-9883

HIV Protease Microbiology/Virology; Proteases/Proteasome
Bictegravir (GS-9883) 是一种 HIV-1 整合酶抑制剂,其IC50值为 7.5 nM。
T13974 ZL0580

Epigenetic Reader Domain; HIV Protease Chromatin/Epigenetic; Microbiology/Virology; Proteases/Proteasome
ZL0580 通过抑制 Tat 反式激活和转录延伸以及通过在 HIV 启动子处诱导抑制性染色质结构来诱导 HIV 抑制。
T0289 9-Aminoacridine

Aminacrine,9-氨基吖啶

Others; HIV Protease; Antibacterial Microbiology/Virology; Others; Proteases/Proteasome
9-Aminoacridine 是一种具有龋齿传播特性的抗菌剂,可用作局部消毒剂。它也是一种高度荧光染料,实验用作一种诱变剂,是细胞内 pH 的指示剂。
T3172 Trovirdine

曲韦定,LY300046

HIV Protease Microbiology/Virology; Proteases/Proteasome
Trovirdine (LY300046) 是一种硫脲类非核苷类逆转录酶抑制剂。
T16098 Islatravir

MK-8591

HIV Protease; Reverse Transcriptase Microbiology/Virology; Proteases/Proteasome
Islatravir (MK-8591) 是一种核苷逆转录酶抑制剂,是抗HIV-1药物,对 HIV-1 (WT),HIV-1 (M184V),HIV-1 (MDR) 的EC50值分别为 0.068 nM,3.1 nM 和 0.15 nM。
T9212 IMB-301

Others; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
IMB-301是根据 hA3G 模型通过虚拟筛选的一种小分子抑制剂。
T4557 Amylmetacresol

戊甲酚,5-Methyl-2-Pentylphenol

Others; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
Amylmetacresol (5-Methyl-2-Pentylphenol) 是一种有潜力研究咽喉痛相关疾病的抗病毒化合物。
T10603 BRD-6929

HIV Protease; HDAC Chromatin/Epigenetic; DNA Damage/DNA Repair; Microbiology/Virology; Proteases/Proteasome
BRD-6929 是一种选择性的脑渗透性的HDAC1和HDAC2抑制剂 ,IC50值为 1 和 8 nM。它对 HDAC1 和 HDAC2 有高亲和力,Ki 值为  0.2 和 1.5 nM。它可研究情绪相关行为。
T15371 Gardiquimod

TLR; HIV Protease Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
Gardiquimod 可抑制巨噬细胞和活化的外周血单个核细胞的HIV-1感染。 它是一种咪唑喹啉类似物,是一种 TLR7/8 激动剂。
T10133 3'-Azido-3'-deoxy-5-methylcytidine

Antiviral; HIV Protease Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
3'-Azido-3'-deoxy-5-methylcytidine 抑制 HIV-1 逆转录酶 (EC50 = 0.06 μM),是异嗜性鼠白血病相关逆转录病毒 (XMRV, CC50 = 43.5 μM) 的有效抑制剂。
T11538 Hck-IN-1

HIV Protease; Src; Hck Angiogenesis; Microbiology/Virology; Proteases/Proteasome; Tyrosine Kinase/Adaptors
Hck-IN-1 是二苯基吡唑啉化合物,选择性的 Nef 依赖性 Hck 抑制剂。它是广泛的 HIV-1 Nef 直接拮抗剂,对于野生型 HIV-1 复制的IC50为 100-300 nM。它结合口袋残基 Asn126,具有抗逆转录病毒活性。
TQ0174 Mavorixafor

AMD-070

CXCR Autophagy; GPCR/G Protein; Immunology/Inflammation
Mavorixafor (AMD-070) 是一种有效的特异性 CXCR4 拮抗剂,对 CXCR4 125I-SDF 结合的 IC50 值为 13 nM。 Mavorixafor 在 MT-4 细胞 (IC50 = 1 nM) 和 PBMC (IC50 = 9 nM) 中抑制 T-tropic HIV-1 (NL4.3 株) 的复制。
T9039 HIV-1 Nef-IN-1

HIV Protease Microbiology/Virology; Proteases/Proteasome
HIV-1 Nef-IN-1 是 HIV-1 Nef 蛋白的抑制剂。 它有效地竞争 Nef-SH3Hck 相互作用,Kd 值为 6.7 μM。
T6846 Vesatolimod

GS-9620,维沙莫德

Apoptosis; HCV Protease; HBV; TLR; HIV Protease Apoptosis; Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
Vesatolimod (GS-9620) 是一种选择性 Toll 样受体 7 口服激动剂,EC50值为291 nM。
T0781 Dimercaprol

Dicaptol,二巯丙醇,Dithiopropanol,二巯基丙醇

Others; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
Dimercaprol (Dicaptol) 是一种具有抗HIV 活性的重金属中毒解毒剂。
T8238 Fosamprenavir Calcium Salt

福沙那伟钙,Diallyl Trisulfide,GW433908G

HIV Protease Microbiology/Virology; Proteases/Proteasome
Fosamprenavir Calcium Salt (GW433908G) 是抗逆转录病毒蛋白酶抑制剂 Amprenavir 的磷酸酯前药,具有改善的溶解性和抗HIV 感染作用。
T6007 Birinapant

TL32711,比瑞那帕

Apoptosis; IAP; HIV Protease Apoptosis; Microbiology/Virology; Proteases/Proteasome
Birinapant (TL32711) 是一种二价 Smac 模拟物,是 XIAP 和 cIAP1的强效拮抗剂,Kd 值分别为 45 nM 和小于 1 nM。它靶向与 TRAF2 相关的 cIAP,并消除 TNF 诱导的 NF-κB 活化。
T10570 Fostemsavir Tris

BMS-663068 Tris

HIV Protease Microbiology/Virology; Proteases/Proteasome
Fostemsavir Tris (BMS-663068 Tris) 是一种 HIV-1附着抑制剂。
T3523 Fostemsavir

BMS-663068,磷坦姆沙韦

HIV Protease Microbiology/Virology; Proteases/Proteasome
Fostemsavir (BMS-663068) 是 BMS-626529 的原药,可抑制 HIV-1 与细胞 CD4 受体的结合,能结合gp120。
T2239L Raltegravir

雷特格韦,MK-0518

HIV Protease; Integrase Microbiology/Virology; Proteases/Proteasome
Raltegravir (MK-0518) 是一种HIV 整合酶抑制剂。
T0033 Miltefosine

HePC,米替福新,Hexadecyl phosphocholine

Akt; HIV Protease; PKC Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology; PI3K/Akt/mTOR signaling; Proteases/Proteasome
Miltefosine (HePC) 是一种广谱抗微生物剂,是治疗内脏和皮肤利什曼病的药物。它是 CTP 磷酸胆碱胞苷基转移酶的抑制剂。
T0753 Salicylanilide

WR10019,2-Hydroxybenzanilide,水杨酰苯胺

HIV Protease; Reverse Transcriptase Microbiology/Virology; Proteases/Proteasome
Salicylanilide (2-Hydroxybenzanilide) 有广泛的生物学特性,如抗病毒、菌和抗真菌活性。
TP1432 Enfuvirtide acetate

醋酸恩夫韦地

HIV Protease Microbiology/Virology; Proteases/Proteasome
Enfuvirtide acetate 是一种抗HIV-1融合的抑制肽,是一种由 36 个氨基酸组成的线性合成肽。 它具有乙酰化的 N 端和羧酰胺 C 端。
T3614 Inosine pranobex

Groprinosin,Isoprinosine,异丙肌苷,Immunovir,Delimmun

IL Receptor; HIV Protease Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
Inosine pranobex (Delimmun) 是一种免疫增强剂,它是一种广谱抗病毒剂,用于 HIV 感染。
T11465 Lenacapavir

GS-6207

Others; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
Lenacapavir (GS-6207) 是一种有效的靶向衣壳的 HIV 复制抑制剂。 Lenacapavir 在 MT-4 细胞中显示出抗 HIV 活性,EC50 为 100 pM。
T4697 ABBV-744

ABBV744

Epigenetic Reader Domain; HIV Protease Chromatin/Epigenetic; Microbiology/Virology; Proteases/Proteasome
ABBV-744 是一种 BDII 选择性 BET 溴结构域抑制剂,可抑制 BRD2/3/4。 它可研究炎症性疾病、癌症和艾滋病。
T7903 Saquinavir

Ro 31-8959,沙奎那韦

SARS-CoV; HIV Protease Microbiology/Virology; Proteases/Proteasome
Saquinavir (Ro 31-8959) 是一种 HIV 蛋白酶抑制剂,可研究逆转录病毒。它也是 SARS-CoV 3CLpro 抑制剂,IC50为 1.36 μM。
T5965 Ditiocarb sodium

Sodium diethyldithiocarbamate,二乙基二硫代氨基甲酸钠

HIV Protease Microbiology/Virology; Proteases/Proteasome
Ditiocarb sodium (Sodium diethyldithiocarbamate) 是一种铜胶结率的促进剂。它可降低HIV 感染。
T0282 Q-VD-OPH

Quinoline-Val-Asp-Difluorophenoxymethylketone

Caspase; HIV Protease Apoptosis; Microbiology/Virology; Proteases/Proteasome
Q-VD-OPH (Quinoline-Val-Asp-Difluorophenoxymethylketone) 是一种具有强效抗凋亡特性的泛半胱天冬酶抑制剂。它可抑制 HIV 感染,能透过血脑屏障。
T1883 Des(benzylpyridyl) Atazanavi

HIV Protease Microbiology/Virology; Proteases/Proteasome
Des(benzylpyridyl) Atazanavi 是 Atazanavir 的 N-脱烷基代谢物 (M1),一种 HIV 蛋白酶抑制剂。
T6255 Bromosporine

Epigenetic Reader Domain; CDK Cell Cycle/Checkpoint; Chromatin/Epigenetic
Bromosporine 是广谱 BRD2/4/9 和 CECR2 溴结构域抑制剂,IC50为0.41、0.29、0.122和0.017 μM。
T0676 Hydroxyurea

Hydroxycarbamide,羟基脲,nsc32065,nci-c04831

Apoptosis; HIV Protease; DNA/RNA Synthesis; Autophagy Apoptosis; Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Proteases/Proteasome
Hydroxyurea (Hydroxycarbamide) 是一种抗肿瘤剂,通过抑制核糖核苷二磷酸还原酶来抑制 DNA 合成。
T16154 MS417

GTPL7512

Epigenetic Reader Domain; HIV Protease Chromatin/Epigenetic; Microbiology/Virology; Proteases/Proteasome
MS417 (GTPL7512) 是一种 BET 特异性 BRD4 抑制剂,与 BRD4-BD1 和 BRD4-BD2 结合,Kd 值分别为 36.1和25.4 nM,IC50值分别为 30和46 nM。它对 CBP BRD 的选择性较低,IC50值为 32.7 μM。
T6214 Emtricitabine

恩曲他滨,FTC,Emtriva,BW1592

HIV Protease; Reverse Transcriptase Microbiology/Virology; Proteases/Proteasome
Emtricitabine (FTC) 是一种核苷逆转录酶抑制剂, 在 PBMC 细胞中的 EC50值为0.01 µM,可研究 HIV 感染。
T1649 Tenofovir

替诺福韦,泰诺福韦,PMPA,TDF,GS 1278

HBV; HIV Protease; Reverse Transcriptase Microbiology/Virology; Proteases/Proteasome
Tenofovir (GS 1278) 是一种核苷酸逆转录酶抑制剂,可研究 HIV 和慢性乙型肝炎。

化合物

TAT
Cat.No: TP1809
Synonym:
Target: HIV Protease
PMEDAP
Cat.No: T38514
Synonym:
Target: Others, HIV Protease
Sodium copper chlorophyllin B
Cat.No: T12953
Synonym:
Target: Influenza Virus, HIV Protease
RN-18
Cat.No: T16764
Synonym:
Target: HIV Protease
GSK2838232
Cat.No: T15436
Synonym:
Target: HIV Protease
3-Deazaadenosine hydrochloride
Cat.No: T10111
Synonym:
Target: Others, HIV Protease
Reverse transcriptase-IN-1
Cat.No: T12715
Synonym:
Target: HIV Protease
Clathrin-IN-1
Cat.No: T9063
Synonym:
Target: HIV Protease
YYA-021
Cat.No: T6256
Synonym: YYA 021
Target: gp120/CD4, HIV Protease
NBD-556
Cat.No: T16276
Synonym:
Target: HIV Protease
Temsavir
Cat.No: T4665
Synonym: BMS626529
Target: HIV Protease
Elsulfavirine
Cat.No: T15210
Synonym: Elpida,VM-1500
Target: HIV Protease
Sulfadoxine
Cat.No: T0836
Synonym: 周效磺胺,磺胺多辛,Sulphadoxine
Target: DHFR, HIV Protease, Antibiotic, Parasite, Autophagy
Probenecid
Cat.No: T0457
Synonym: Benemid,丙磺舒
Target: HIV Protease, Antibacterial, TRP/TRPV Channel
Obefazimod
Cat.No: T8311
Synonym: ABX-464,ABX464
Target: HIV Protease
Bictegravir
Cat.No: T4493
Synonym: GS-9883
Target: HIV Protease
ZL0580
Cat.No: T13974
Synonym:
Target: Epigenetic Reader Domain, HIV Protease
9-Aminoacridine
Cat.No: T0289
Synonym: Aminacrine,9-氨基吖啶
Target: Others, HIV Protease, Antibacterial
Trovirdine
Cat.No: T3172
Synonym: 曲韦定,LY300046
Target: HIV Protease
Islatravir
Cat.No: T16098
Synonym: MK-8591
Target: HIV Protease, Reverse Transcriptase
IMB-301
Cat.No: T9212
Synonym:
Target: Others, HIV Protease
Amylmetacresol
Cat.No: T4557
Synonym: 戊甲酚,5-Methyl-2-Pentylphenol
Target: Others, HIV Protease
BRD-6929
Cat.No: T10603
Synonym:
Target: HIV Protease, HDAC
Gardiquimod
Cat.No: T15371
Synonym:
Target: TLR, HIV Protease
3'-Azido-3'-deoxy-5-methylcytidine
Cat.No: T10133
Synonym:
Target: Antiviral, HIV Protease
Hck-IN-1
Cat.No: T11538
Synonym:
Target: HIV Protease, Src, Hck
Mavorixafor
Cat.No: TQ0174
Synonym: AMD-070
Target: CXCR
HIV-1 Nef-IN-1
Cat.No: T9039
Synonym:
Target: HIV Protease
Vesatolimod
Cat.No: T6846
Synonym: GS-9620,维沙莫德
Target: Apoptosis, HCV Protease, HBV, TLR, HIV Protease
Dimercaprol
Cat.No: T0781
Synonym: Dicaptol,二巯丙醇,Dithiopropanol,二巯基丙醇
Target: Others, HIV Protease
Fosamprenavir Calcium Salt
Cat.No: T8238
Synonym: 福沙那伟钙,Diallyl Trisulfide,GW433908G
Target: HIV Protease
Birinapant
Cat.No: T6007
Synonym: TL32711,比瑞那帕
Target: Apoptosis, IAP, HIV Protease
Fostemsavir Tris
Cat.No: T10570
Synonym: BMS-663068 Tris
Target: HIV Protease
Fostemsavir
Cat.No: T3523
Synonym: BMS-663068,磷坦姆沙韦
Target: HIV Protease
Raltegravir
Cat.No: T2239L
Synonym: 雷特格韦,MK-0518
Target: HIV Protease, Integrase
Miltefosine
Cat.No: T0033
Synonym: HePC,米替福新,Hexadecyl phosphocholine
Target: Akt, HIV Protease, PKC
Salicylanilide
Cat.No: T0753
Synonym: WR10019,2-Hydroxybenzanilide,水杨酰苯胺
Target: HIV Protease, Reverse Transcriptase
Enfuvirtide acetate
Cat.No: TP1432
Synonym: 醋酸恩夫韦地
Target: HIV Protease
Inosine pranobex
Cat.No: T3614
Synonym: Groprinosin,Isoprinosine,异丙肌苷,Immunovir,Delimmun
Target: IL Receptor, HIV Protease
Lenacapavir
Cat.No: T11465
Synonym: GS-6207
Target: Others, HIV Protease
ABBV-744
Cat.No: T4697
Synonym: ABBV744
Target: Epigenetic Reader Domain, HIV Protease
Saquinavir
Cat.No: T7903
Synonym: Ro 31-8959,沙奎那韦
Target: SARS-CoV, HIV Protease
Ditiocarb sodium
Cat.No: T5965
Synonym: Sodium diethyldithiocarbamate,二乙基二硫代氨基甲酸钠
Target: HIV Protease
Q-VD-OPH
Cat.No: T0282
Synonym: Quinoline-Val-Asp-Difluorophenoxymethylketone
Target: Caspase, HIV Protease
Des(benzylpyridyl) Atazanavi
Cat.No: T1883
Synonym:
Target: HIV Protease
Bromosporine
Cat.No: T6255
Synonym:
Target: Epigenetic Reader Domain, CDK
Hydroxyurea
Cat.No: T0676
Synonym: Hydroxycarbamide,羟基脲,nsc32065,nci-c04831
Target: Apoptosis, HIV Protease, DNA/RNA Synthesis, Autophagy
MS417
Cat.No: T16154
Synonym: GTPL7512
Target: Epigenetic Reader Domain, HIV Protease
Emtricitabine
Cat.No: T6214
Synonym: 恩曲他滨,FTC,Emtriva,BW1592
Target: HIV Protease, Reverse Transcriptase
Tenofovir
Cat.No: T1649
Synonym: 替诺福韦,泰诺福韦,PMPA,TDF,GS 1278
Target: HBV, HIV Protease, Reverse Transcriptase
Cat. No. Product Name Target Signaling Pathways
T6377 Aloperine

Apoptosis; Virus Protease; HIV Protease; Antibiotic; Autophagy Apoptosis; Autophagy; Microbiology/Virology; Proteases/Proteasome
Aloperine 是一种在苦参类植物中的生物碱,其具有抗癌,抗炎、抗肿瘤和抗病毒特性,可用于研究过敏性接触性皮炎湿疹和其他皮肤炎症。
TN2283 Tripterifordin

HIV Protease Microbiology/Virology; Proteases/Proteasome
Tripterifordin 在 H9 淋巴细胞中显示出抗 HIV 复制活性,EC50值为 3100 nM。
TQ0217 Gomisin G

戈米辛G,戈米辛 G

P450; HIV Protease Metabolism; Microbiology/Virology; Proteases/Proteasome
Gomisin G 是一种有抗HIV 活性的天然产物。
T2942 Psoralen

Ficusin,Furocoumarin,补骨脂素,psoralene

Apoptosis; Influenza Virus; HIV Protease; DNA/RNA Synthesis Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Proteases/Proteasome
Psoralen (Ficusin) 是从补骨脂种子中提取的一种香豆素。它具有如抗癌、抗氧化、抗抑郁、抗癌、抗菌、抗病毒等多种生物学特性。
TN1103 Diphyllin

山荷叶素,二叶草素

ATPase; Proton pump; Influenza Virus; HIV Protease Membrane transporter/Ion channel; Microbiology/Virology; Proteases/Proteasome
Diphyllin 是一种从Justicia procumbens 中分离的芳基萘木脂素,是HIV-1的有效抑制剂,IC50 为 0.38 μM。它是V-ATPase 抑制剂,IC50值为 17 nM,可抑制人破骨细胞中的溶酶体酸化。它抑制NO 产生,IC50值为 50 μM ,具有抗癌和抗炎活性。
T0474 Erythromycin ethylsuccinate

EES,琥乙红霉素

ribosome; HIV Protease; Antibacterial; Antibiotic; Autophagy Autophagy; Microbiology/Virology; Proteases/Proteasome
Erythromycin ethylsuccinate (EES) 是一种由红链霉菌产生的大环内酯类抗生素,有潜力用于多种细菌感染。它具有抗 HIV-1病毒活性。
Fr16741 Oxindole

2-吲哚酮,板蓝根,Indolin-2-one

Others; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
Oxindole (Indolin-2-one) 是一种芳族杂环砌块,其衍生物是激酶抑制剂研究中的主要成分。
T2865 Oleanolic Acid

Oleanic acid,Caryophyllin,齐墩果酸

HIV Protease; Endogenous Metabolite; Antibiotic; Autophagy Autophagy; Metabolism; Microbiology/Virology; Proteases/Proteasome
Oleanolic Acid (Caryophyllin) 是具有抗癌活性的一种天然产物。
T3822 Bellidifolin

Bellidifoline,龙胆山酮酚,Bellidifolium,雏菊叶龙胆酮

Others; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
Bellidifolin (Bellidifoline) 是从獐牙菜的茎中提取的一种呫吨酮,它能作为病毒蛋白 R 的抑制剂,具有保肝、降血糖、抗炎、抗氧化、抗肿瘤作用。
T0966 Sennoside A

番泻苷A,NSC 112929,番泻苷 A

MAO; HIV Protease Metabolism; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Sennoside A (NSC-112929) 是在番泻叶的叶子和豆荚中大量发现的蒽醌苷,抑制 HIV-1 复制。
T6841 Fumagillin

NSC9168,烟曲霉素,Amebacilin

Others; HIV Protease; Antibiotic; Parasite Microbiology/Virology; Others; Proteases/Proteasome
Fumagillin (Amebacilin) 由烟曲霉菌中提取的一种抗菌药,有抗阿米巴活性。它通过抑制 HIV-1 viral protein R 活性来抑制 HIV‐1感染。
T1131 Ivermectin

MK-933,伊维菌素

Mitophagy; GluCls; P2X Receptor; SARS-CoV; HIV Protease; Antibiotic; Parasite; Autophagy; HSV Autophagy; Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Ivermectin (MK-933) 是谷氨酸门控氯离子通道激活剂,具有抗寄生虫活性。它特异性抑制Impα/β1 介导的核导入,还抑制牛疱疹病毒 1 复制并抑制BoHV-1DNA 聚合酶的核输入。它具有很强的抗病毒活性。它也是P2X4和 α7nAChRs 的正异构效应物。
T8116 Azulene

甘菊蓝,奥苷菊环,Bicyclo[5.3.0]Decapentaene

Others; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
Azulene (Bicyclo[5.3.0]Decapentaene) 是萘的异构体,具有高抗HIV 活性。它是从洋甘菊精油中分离出来的一种化学支架。
T8689 Chloroquine

CQ,氯喹

SARS-CoV; TLR; HIV Protease; Antibiotic; Parasite; Autophagy Autophagy; Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
Chloroquine 是一种 Toll 样受体抑制剂,可以抑制自噬。Chloroquine 具有抗疟疾和抗炎活性,广泛用于治疗疟疾和类风湿性关节炎。Chloroquine 还具有抗 SARS-CoV-2 (COVID-19) 活性、抗 HIV-1 活性。
T2177 Kaempferol

Kempferol,山柰酚,山奈酚,Robigenin

Apoptosis; Estrogen Receptor/ERR; Mitophagy; Estrogen/progestogen Receptor; HIV Protease; Endogenous Metabolite; Parasite; Autophagy Apoptosis; Autophagy; Endocrinology/Hormones; Metabolism; Microbiology/Virology; Proteases/Proteasome
Kaempferol (Robigenin) 属于天然类黄酮,是一种 ERRα 和 ERRγ 的反向激动剂。Kaempferol 具有抗肿瘤、抗炎、抗氧化、抗菌和抗病毒等多种活性。
T2S0731 Trilobatin

三叶苷,三叶甙,P-Phlorizin

Amylase Metabolism
Trilobatin (P-Phlorizin) 是源自Lithocarpus polystachyusRehd 的甜味剂,是一种HIV-1抑制剂,靶向 Gp41 包膜蛋白,具有神经保护作用。它还是SGLT1/2抑制剂,可选择性诱导人肝母细胞瘤细胞增殖。
T0492 Dimethyl fumarate

富马酸二甲酯,DMF

Reactive Oxygen Species; HIV Protease; Nrf2; Endogenous Metabolite; Autophagy Autophagy; Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
Dimethyl fumarate (DMF) 是具有口服活性且可透过血脑屏障的Nrf2激活剂,可诱导抗氧化剂基因表达上调。它是一种富马酸盐衍生物,可作抗炎和免疫调节剂,可研究多发性硬化症。
T4962 Zingibroside R1

Ginsenoside Z-R1,姜状三七皂苷R1,姜状三七苷R1

HIV Protease Microbiology/Virology; Proteases/Proteasome
Zingibroside R1 (Ginsenoside Z-R1) 是分离自Panax japonicasC. A. Meyer 根部的一种三萜皂苷,有HIV-1、抗肿瘤和抗血管生成活性。它对 EAT 细胞的 2-脱氧-D-葡萄糖的摄取具有抑制作用,IC50值为91.3 μM。
T2789 Scutellarin

黄岑素,野黄芩苷,Breviscapin,Breviscapinun,Breviscapine,Scutellarein-7-glucuronide

Akt; HIV Protease; STAT Cytoskeletal Signaling; JAK/STAT signaling; Microbiology/Virology; PI3K/Akt/mTOR signaling; Proteases/Proteasome; Stem Cells
Scutellarin (Scutellarein-7-glucuronide) 是从黄芩中分离的黄酮,可抑制破骨细胞中 RANKL 介导的 MAPK 和 NF-κB 信号通路,并下调 HCC 细胞中的 STAT3/Girdin/Akt 信号通路。
T2728 Limonin

Dictamnolactone,Limonoic acid 3,19:16,17 dilactone,柠檬苦素,Obaculactone,Citrolimonin

Apoptosis; HIV Protease; Endogenous Metabolite Apoptosis; Metabolism; Microbiology/Virology; Proteases/Proteasome
Limonin (Citrolimonin) 是柑橘类水果中富含的一种三萜类天然产物,具有抗病毒和抗肿瘤活性。
T5429 Theaflavin 3,3'-digallate

茶黄素-3,3'-双没食子酸,8-Gingerol,TFDG

Virus Protease; Antioxidant; HIV Protease; HSV Microbiology/Virology; oxidation-reduction; Proteases/Proteasome
Theaflavin 3,3'-digallate (8-Gingerol) 是一种寨卡病毒蛋白酶抑制剂,IC50为 2.3 μM。它直接与 ZIKVpro 结合并抑制 ZIKV 复制,可抑制 gp41 和 NS2B-3 蛋白酶的活性,并具有抗 HSV 和 HIV-1病毒活性。它是红茶中的主要多酚,有抗肿瘤作用。
T1284 Megestrol acetate

SC10363,醋酸甲地孕酮,BDH1298

Glucocorticoid Receptor; Estrogen/progestogen Receptor; Progesterone Receptor; HIV Protease; Autophagy Autophagy; Endocrinology/Hormones; Microbiology/Virology; Others; Proteases/Proteasome
Megestrol acetate (BDH1298) 是具有口服活性的合成孕激素。它还具有抗雄激素特性,可用于治疗厌食症和恶病质。
T7991 2-Hydroxycinnamic acid

邻羟基肉桂酸(邻香豆酸),(E)-3-(2-羟基苯基)丙烯酸

Others; SARS-CoV; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
2-Hydroxycinnamic acid 是从肉桂的甲醇提取物中分离出的一种天然产物,具有光氧化活性。它对HIV/SARS-CoV S 假病毒的感染具有抑制作用,IC50为 0.3 mM。
T16791 Rottlerin

Mallotoxin,NSC 56346,粗糠柴苦素,NSC 94525

CaMK; Apoptosis; Others; HIV Protease; PKA; PKC; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology; Neuroscience; Others; Proteases/Proteasome; Tyrosine Kinase/Adaptors
Rottlerin (NSC-56346) 是一种从Mallotus Philippinensis 中得到的天然产物, 是 PKC 的特异性抑制剂,抑制HIV-1整合和狂犬病病毒感染。它通过活化 caspase 3 诱导细胞凋亡.
T3122 Fangchinoline

Tetrandrine B,防己诺林碱,(+)-Limacine,Hanfangichin B,防己醇灵,(+)-Fangchinoline

Apoptosis; FAK; HIV Protease; Autophagy Angiogenesis; Apoptosis; Autophagy; Cytoskeletal Signaling; Microbiology/Virology; Proteases/Proteasome; Tyrosine Kinase/Adaptors
Fangchinoline (Tetrandrine B) 是从Stephaniatetrandra 中分离出来的,一种具有广泛生物学活性的天然产物。它是新型HIV-1抑制剂,通过损害 gp160 蛋白水解过程来抑制 HIV-1 复制。它靶向Focal adhesion kinase (FAK)并抑制肿瘤细胞中 FAK 介导的的信号传导途径。
T3730 Methyl gallate

NSC 363001,Gallicin,Gallic acid methyl ester,Gallincin,没食子酸甲酯

Reactive Oxygen Species; HIV Protease; Reverse Transcriptase; Antibacterial Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
Methyl gallate (Gallincin) 是具有抗氧化,抗癌和抗炎活性的植物酚类。它也可抑制细菌活性。它还具有抗HIV-1和HIV-1酶的抑制活性。
T2775 Baicalin

黄芩苷,黄岑苷,Baicalein 7-O-β-D-glucuronide

NF-κB; HIV Protease; GABA Receptor; Autophagy Autophagy; Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience; NF-κB; Proteases/Proteasome
Baicalin (Baicalein 7-O-β-D-glucuronide) 是一种从黄芩中分离出来的脯氨酰内肽酶抑制剂,具有抗氧化、抗肿瘤、抗 HIV 的特性。
T1020 Doxorubicin hydrochloride

Adriamycin,Doxorubicin (Adriamycin) HCl,Hydroxydaunorubicin hydrochloride,盐酸多柔比星,盐酸阿霉素,NSC 123127

Apoptosis; Mitophagy; HBV; HIV Protease; Topoisomerase; Antibacterial; Antibiotic; AMPK; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair; Microbiology/Virology; PI3K/Akt/mTOR signaling; Proteases/Proteasome
Doxorubicin hydrochloride (Adriamycin) 属于蒽环类抗生素,是人类 DNA 拓扑异构酶 I/II 抑制剂 (IC50=0.8/2.67 μM)。Doxorubicin hydrochloride 具有细胞毒性和抗肿瘤活性。Doxorubicin hydrochloride 可降低 AMPK 及其下游靶蛋白乙酰辅酶 A 羧化酶的磷酸化,还可诱导凋亡和自噬。
T2830 Betulinic acid

白桦脂酸,桦木酸,ALS-357,Lupatic acid,Betulic acid

Apoptosis; Mitophagy; NF-κB; HIV Protease; Topoisomerase; Endogenous Metabolite; Aminopeptidase; Autophagy Apoptosis; Autophagy; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
Betulinic acid (ALS-357) 是从白桦树皮中分离出来的一种五环三萜类天然产物,是真核细胞拓扑异构酶 I 的抑制剂,IC50值为 5 μM,具有抗逆转录病毒、抗疟疾、抗癌和抗炎特性。
T5782 Bevirimat

YK FH312,MPC-4326,PA-457,贝韦立马

HIV Protease Microbiology/Virology; Proteases/Proteasome
Bevirimat (PA-457) 是一种 HIV-1 成熟抑制剂,可在病毒体成熟过程中阻断 Gag 衣壳 (CA) 前体 CA-SPI 裂解为成熟的 CA 蛋白。
T0194 Chloroquine phosphate

Chloroquine diphosphate,Aralen phosphate,磷酸氯喹,Chingamin phosphate

SARS-CoV; TLR; HIV Protease; Antibiotic; Parasite; Autophagy Autophagy; Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
Chloroquine phosphate (Aralen phosphate) 是广泛用于疟疾和类风湿性关节炎的抗疟疾和抗炎剂。它是autophagy 和toll-like receptors 抑制剂,有效抑制SARS-CoV-2(COVID-19) 感染 (EC50=1.13 μM)。
T3772 Maslinic acid

2α-Hydroxyoleanoic Acid,山楂酸,2α-Hydroxyoleanolic acid,Crategolic acid

NF-κB; HIV Protease; DNA/RNA Synthesis; Antibacterial Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; NF-κB; Proteases/Proteasome
Maslinic acid (Crategolic acid) 是一种 DNA 聚合酶 B 抑制剂,抑制 NF-κB p65的 DNA 结合活性并消除 IκB-α磷酸化。
T6S2391 L-Chicoric Acid

(-)-Chicoric acid,trans-Caffeoyltartaric acid,Chicoric acid,L-菊苣酸,dicaffeoyltartaric acid,菊苣酸

Others; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
L-Chicoric Acid (trans-Caffeoyltartaric acid) 是一种二咖啡酰酒石酸,是一种选择性可逆的 HIV-1 整合酶抑制剂,IC50约为 100 nM。它还可抑制 HIV-1 复制。
T0070 Pentoxifylline

Oxpentifylline,PTX,己酮可可碱,BL-191

HIV Protease; PDE; Adenosine Receptor; Autophagy Autophagy; GPCR/G Protein; Metabolism; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Pentoxifylline (PTX) 是一种具有口服活性的磷酸二酯酶非选择性抑制剂,具有免疫调节、抗炎、抗纤溶、抗增殖和血液流变学改善作用。它可研究周围血管疾病、脑血管疾病和其他一些涉及局部微循环缺陷的疾病。
T0710 L-Cycloserine

Levcycloserine,Levcicloserina,(-)-Cycloserine,(S)-Cycloserine,Levcycloserinum,环丝氨酸,(S)-4-Amino-3-isoxazolidone

HIV Protease; GABA Receptor Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience; Proteases/Proteasome
L-Cycloserine ((-)-Cycloserine) 不可逆地抑制大肠杆菌以及各种动物大脑中的 GABA 吡哆醛 5'-磷酸依赖性转氨酶,导致体内抑制性神经递质 γ-氨基丁酸水平升高。
T3321 Oleanonic acid

3-Oxooleanolic acid,3-Oxoolean-12-en-28-oic Acid,Oleanonic Acid,齐墩果酮酸,3-Ketooleanolic Acid

HIV Protease Microbiology/Virology; Proteases/Proteasome
Oleanonic acid (3-Ketooleanolic Acid) 是一种三萜,可以抑制 HIV-1 对细胞的感染。它具有保肝作用,并具有抗肿瘤和抗病毒特性。
T1125 Shikonin

NSC 252844,Isoarnebin 4,(+)-Shikonin,紫草素,Alkanna Red,C.I. 75535,Anchusa acid

TNF; NF-κB; Chloride channel; HIV Protease; PKM Apoptosis; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
Shikonin (Anchusa acid) 属于天然产物,是一种 TMEM16A 氯离子通道抑制剂 (IC50=6.5 μM) 和选择性 PKM2 抑制剂。Shikonin 具有抗肿瘤、抗炎和伤口愈合活性。
T22468 1-Deoxymannojirimycin hydrochloride

Others; Influenza Virus; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
1-Deoxymannojirimycin hydrochloride 是一种选择性的 α1,2-甘露糖苷酶抑制剂,IC50值为 20 μM。它还抑制 HIV-1 毒株,抗病毒活性较差。
T7064 Valproic Acid

Sodium valproate,2-Propylpentanoic Acid,丙戊酸,VPA,Depakine,2-Propylvaleric Acid

Mitophagy; Gamma-secretase; HIV Protease; GABA Receptor; Sodium Channel; HDAC; Autophagy Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience; Proteases/Proteasome; Stem Cells
Valproic Acid (2-Propylpentanoic Acid) 是一种 HDAC 抑制剂,可抑制 HDAC1 活性,诱导 HDAC2 降解,具有口服活性。Valproic Acid 可以用于癫痫和躁郁症的研究。
T0200 α-Lipoic Acid

Thioctic acid,DL-α-Lipoic acid,(±)-α-Lipoic acid,α-硫辛酸,硫辛酸

Apoptosis; NF-κB; HIV Protease; Mitochondrial Metabolism; Endogenous Metabolite Apoptosis; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
α-Lipoic Acid (DL-α-Lipoic acid) 是线粒体酶复合物的重要辅助因子,是一种抗氧化剂,可抑制NF-κB 依赖性的HIV-1LTR 活化。它还可诱导内质网应激介导的肝癌细胞凋亡。
T1456 Doxorubicin

Hydroxydaunorubicin,阿霉素,Adriamycin

Topoisomerase; AMPK Chromatin/Epigenetic; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
Doxorubicin (Adriamycin) 是一种有细胞毒性的蒽环类抗生素,具有肿瘤化疗作用。它抑制DNA 拓扑异构酶 I 和拓扑异构酶 II,IC50分别为0.8 μM 和2.67 μM,从而抑制 DNA 复制。它下调AMPK 的基础磷酸化以及下游 acetyl-CoA 羧化酶。它诱导凋亡和自噬 。
T5783 Rosamultin

野蔷薇苷,罗莎白素

Antioxidant; HIV Protease Microbiology/Virology; oxidation-reduction; Proteases/Proteasome
Rosamultin 是从Potentilla anserina L 分离的 19 α-羟基型三萜。它抑制 HIV-1 蛋白酶,具有抗氧化、抗炎和镇痛作用。
T4537 Cholic acid sodium

胆酸钠,[胆酸钠],SodiumCholate

HIV Protease; Endogenous Metabolite Metabolism; Microbiology/Virology; Proteases/Proteasome
Cholic acid sodium (SodiumCholate) 是肝脏中产生的主要胆汁酸,通常与牛磺酸或甘氨酸结合,有助于脂肪吸收和胆固醇排泄。
TL0006 Cichoric Acid

菊苣酸,Dicaffeoyltartaric acid,Chicoric Acid

Reactive Oxygen Species; HIV Protease Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
Cichoric Acid (Dicaffeoyltartaric acid) 是一种天然化合物,具有抗氧化作用。
TN2231 Soyasaponin II

Influenza Virus; HIV Protease; HSV Microbiology/Virology; Proteases/Proteasome
Soyasaponin II has antiviral effects, it can inhibit the replication of human cytomegalovirus, influenza virus, and human immunodeficiency virus type 1.
TN4109 Ganolucidic acid A

HIV Protease Microbiology/Virology; Proteases/Proteasome
Ganolucidic acid A exhibits cytotoxicity, has inhibitory activities against human HeLa cervical cancer cell lines. It shows significant anti-human immunodeficiency virus (anti-HIV)-1 protease activity with IC50 values of 20-90 microM.
TMA1012 Ganoderiol F

Androgen Receptor; HIV Protease; Autophagy Autophagy; Endocrinology/Hormones; Microbiology/Virology; Proteases/Proteasome
Ganoderiol F has anti-inflammatory, cytotoxic and anti-HIV activity, it inhibits activity of topoisomerases in vitro, and it inhibits human immunodeficiency virus-1 protease with IC(50) values of 20-40 microM. It induced HO-1 expression, activation of the mitogen-activated protein kinase EKR and up-regulation of cyclin-dependent kinase inhibitor p16 and suppressed lipopolysaccharide (LPS)-induced nitric oxide (NO) production.

天然产物

Aloperine
Cat.No: T6377
Synonym:
Target: Apoptosis, Virus Protease, HIV Protease, Antibiotic, Autophagy
Tripterifordin
Cat.No: TN2283
Synonym:
Target: HIV Protease
Gomisin G
Cat.No: TQ0217
Synonym: 戈米辛G,戈米辛 G
Target: P450, HIV Protease
Psoralen
Cat.No: T2942
Synonym: Ficusin,Furocoumarin,补骨脂素,psoralene
Target: Apoptosis, Influenza Virus, HIV Protease, DNA/RNA Synthesis
Diphyllin
Cat.No: TN1103
Synonym: 山荷叶素,二叶草素
Target: ATPase, Proton pump, Influenza Virus, HIV Protease
Erythromycin ethylsuccinate
Cat.No: T0474
Synonym: EES,琥乙红霉素
Target: ribosome, HIV Protease, Antibacterial, Antibiotic, Autophagy
Oxindole
Cat.No: Fr16741
Synonym: 2-吲哚酮,板蓝根,Indolin-2-one
Target: Others, HIV Protease
Oleanolic Acid
Cat.No: T2865
Synonym: Oleanic acid,Caryophyllin,齐墩果酸
Target: HIV Protease, Endogenous Metabolite, Antibiotic, Autophagy
Bellidifolin
Cat.No: T3822
Synonym: Bellidifoline,龙胆山酮酚,Bellidifolium,雏菊叶龙胆酮
Target: Others, HIV Protease
Sennoside A
Cat.No: T0966
Synonym: 番泻苷A,NSC 112929,番泻苷 A
Target: MAO, HIV Protease
Fumagillin
Cat.No: T6841
Synonym: NSC9168,烟曲霉素,Amebacilin
Target: Others, HIV Protease, Antibiotic, Parasite
Ivermectin
Cat.No: T1131
Synonym: MK-933,伊维菌素
Target: Mitophagy, GluCls, P2X Receptor, SARS-CoV, HIV Protease, Antibiotic, Parasite, Autophagy, HSV
Azulene
Cat.No: T8116
Synonym: 甘菊蓝,奥苷菊环,Bicyclo[5.3.0]Decapentaene
Target: Others, HIV Protease
Chloroquine
Cat.No: T8689
Synonym: CQ,氯喹
Target: SARS-CoV, TLR, HIV Protease, Antibiotic, Parasite, Autophagy
Kaempferol
Cat.No: T2177
Synonym: Kempferol,山柰酚,山奈酚,Robigenin
Target: Apoptosis, Estrogen Receptor/ERR, Mitophagy, Estrogen/progestogen Receptor, HIV Protease, Endogenous Metabolite, Parasite, Autophagy
Trilobatin
Cat.No: T2S0731
Synonym: 三叶苷,三叶甙,P-Phlorizin
Target: Amylase
Dimethyl fumarate
Cat.No: T0492
Synonym: 富马酸二甲酯,DMF
Target: Reactive Oxygen Species, HIV Protease, Nrf2, Endogenous Metabolite, Autophagy
Zingibroside R1
Cat.No: T4962
Synonym: Ginsenoside Z-R1,姜状三七皂苷R1,姜状三七苷R1
Target: HIV Protease
Scutellarin
Cat.No: T2789
Synonym: 黄岑素,野黄芩苷,Breviscapin,Breviscapinun,Breviscapine,Scutellarein-7-glucuronide
Target: Akt, HIV Protease, STAT
Limonin
Cat.No: T2728
Synonym: Dictamnolactone,Limonoic acid 3,19:16,17 dilactone,柠檬苦素,Obaculactone,Citrolimonin
Target: Apoptosis, HIV Protease, Endogenous Metabolite
Theaflavin 3,3'-digallate
Cat.No: T5429
Synonym: 茶黄素-3,3'-双没食子酸,8-Gingerol,TFDG
Target: Virus Protease, Antioxidant, HIV Protease, HSV
Megestrol acetate
Cat.No: T1284
Synonym: SC10363,醋酸甲地孕酮,BDH1298
Target: Glucocorticoid Receptor, Estrogen/progestogen Receptor, Progesterone Receptor, HIV Protease, Autophagy
2-Hydroxycinnamic acid
Cat.No: T7991
Synonym: 邻羟基肉桂酸(邻香豆酸),(E)-3-(2-羟基苯基)丙烯酸
Target: Others, SARS-CoV, HIV Protease
Rottlerin
Cat.No: T16791
Synonym: Mallotoxin,NSC 56346,粗糠柴苦素,NSC 94525
Target: CaMK, Apoptosis, Others, HIV Protease, PKA, PKC, Autophagy
Fangchinoline
Cat.No: T3122
Synonym: Tetrandrine B,防己诺林碱,(+)-Limacine,Hanfangichin B,防己醇灵,(+)-Fangchinoline
Target: Apoptosis, FAK, HIV Protease, Autophagy
Methyl gallate
Cat.No: T3730
Synonym: NSC 363001,Gallicin,Gallic acid methyl ester,Gallincin,没食子酸甲酯
Target: Reactive Oxygen Species, HIV Protease, Reverse Transcriptase, Antibacterial
Baicalin
Cat.No: T2775
Synonym: 黄芩苷,黄岑苷,Baicalein 7-O-β-D-glucuronide
Target: NF-κB, HIV Protease, GABA Receptor, Autophagy
Doxorubicin hydrochloride
Cat.No: T1020
Synonym: Adriamycin,Doxorubicin (Adriamycin) HCl,Hydroxydaunorubicin hydrochloride,盐酸多柔比星,盐酸阿霉素,NSC 123127
Target: Apoptosis, Mitophagy, HBV, HIV Protease, Topoisomerase, Antibacterial, Antibiotic, AMPK, Autophagy
Betulinic acid
Cat.No: T2830
Synonym: 白桦脂酸,桦木酸,ALS-357,Lupatic acid,Betulic acid
Target: Apoptosis, Mitophagy, NF-κB, HIV Protease, Topoisomerase, Endogenous Metabolite, Aminopeptidase, Autophagy
Bevirimat
Cat.No: T5782
Synonym: YK FH312,MPC-4326,PA-457,贝韦立马
Target: HIV Protease
Chloroquine phosphate
Cat.No: T0194
Synonym: Chloroquine diphosphate,Aralen phosphate,磷酸氯喹,Chingamin phosphate
Target: SARS-CoV, TLR, HIV Protease, Antibiotic, Parasite, Autophagy
Maslinic acid
Cat.No: T3772
Synonym: 2α-Hydroxyoleanoic Acid,山楂酸,2α-Hydroxyoleanolic acid,Crategolic acid
Target: NF-κB, HIV Protease, DNA/RNA Synthesis, Antibacterial
L-Chicoric Acid
Cat.No: T6S2391
Synonym: (-)-Chicoric acid,trans-Caffeoyltartaric acid,Chicoric acid,L-菊苣酸,dicaffeoyltartaric acid,菊苣酸
Target: Others, HIV Protease
Pentoxifylline
Cat.No: T0070
Synonym: Oxpentifylline,PTX,己酮可可碱,BL-191
Target: HIV Protease, PDE, Adenosine Receptor, Autophagy
L-Cycloserine
Cat.No: T0710
Synonym: Levcycloserine,Levcicloserina,(-)-Cycloserine,(S)-Cycloserine,Levcycloserinum,环丝氨酸,(S)-4-Amino-3-isoxazolidone
Target: HIV Protease, GABA Receptor
Oleanonic acid
Cat.No: T3321
Synonym: 3-Oxooleanolic acid,3-Oxoolean-12-en-28-oic Acid,Oleanonic Acid,齐墩果酮酸,3-Ketooleanolic Acid
Target: HIV Protease
Shikonin
Cat.No: T1125
Synonym: NSC 252844,Isoarnebin 4,(+)-Shikonin,紫草素,Alkanna Red,C.I. 75535,Anchusa acid
Target: TNF, NF-κB, Chloride channel, HIV Protease, PKM
1-Deoxymannojirimycin hydrochloride
Cat.No: T22468
Synonym:
Target: Others, Influenza Virus, HIV Protease
Valproic Acid
Cat.No: T7064
Synonym: Sodium valproate,2-Propylpentanoic Acid,丙戊酸,VPA,Depakine,2-Propylvaleric Acid
Target: Mitophagy, Gamma-secretase, HIV Protease, GABA Receptor, Sodium Channel, HDAC, Autophagy
α-Lipoic Acid
Cat.No: T0200
Synonym: Thioctic acid,DL-α-Lipoic acid,(±)-α-Lipoic acid,α-硫辛酸,硫辛酸
Target: Apoptosis, NF-κB, HIV Protease, Mitochondrial Metabolism, Endogenous Metabolite
Doxorubicin
Cat.No: T1456
Synonym: Hydroxydaunorubicin,阿霉素,Adriamycin
Target: Topoisomerase, AMPK
Rosamultin
Cat.No: T5783
Synonym: 野蔷薇苷,罗莎白素
Target: Antioxidant, HIV Protease
Cholic acid sodium
Cat.No: T4537
Synonym: 胆酸钠,[胆酸钠],SodiumCholate
Target: HIV Protease, Endogenous Metabolite
Cichoric Acid
Cat.No: TL0006
Synonym: 菊苣酸,Dicaffeoyltartaric acid,Chicoric Acid
Target: Reactive Oxygen Species, HIV Protease
Soyasaponin II
Cat.No: TN2231
Synonym:
Target: Influenza Virus, HIV Protease, HSV
Ganolucidic acid A
Cat.No: TN4109
Synonym:
Target: HIV Protease
Ganoderiol F
Cat.No: TMA1012
Synonym:
Target: Androgen Receptor, HIV Protease, Autophagy
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